发明名称 |
PROCESS FOR THE SYNTHESIS OF TELAPREVIR, OR PHARMACEUTICALLY ACCEPTABLE SALTS OR SOLVATES AS WELL AS INTERMEDIATE PRODUCTS THEREOF |
摘要 |
<p>The invention relates to a process for the preparation of telaprevir, or a pharmaceutically acceptable salt or solvate thereof, wherein the process requires a smaller number of process steps and/or does not require the use of toxic and instable compounds compared to the known processes. Another embodiment refers to telaprevir, or a pharmaceutically acceptable salt or solvate thereof as well as to intermediate products for preparation of the same, wherein the afore-mentioned products are obtained by the process described herein.</p> |
申请公布号 |
WO2013135870(A1) |
申请公布日期 |
2013.09.19 |
申请号 |
WO2013EP55397 |
申请日期 |
2013.03.15 |
申请人 |
SANDOZ AG |
发明人 |
FELZMANN, WOLFGANG;BRUNNER, STEFANIE;WILHELM, THORSTEN |
分类号 |
C07D403/12 |
主分类号 |
C07D403/12 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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