发明名称 SUBSTITUTED AZAINDAZOLE COMPOUNDS
摘要 Disclosed are azaindazole compounds of Formula (I): or pharmaceutically acceptable salts thereof, wherein: Q is: (i) 5-membered heteroaryl comprising at least one nitrogen heteroatom and substituted with zero to 2 Rg; or (ii) 9- to 10-membered bicyclic heteroaryl selected from Formula (II) and; wherein Ring A is a 5- to 6-membered aryl or heteroaryl fused ring substituted with zero to 2 Rg; and R1, R2, R3, and Rg are defined herein. Also disclosed are methods of using such compounds in the treatment of at least one CYP17 associated condition, such as, for example, cancer, and pharmaceutical compositions comprising such compounds.
申请公布号 EP2638041(A1) 申请公布日期 2013.09.18
申请号 EP20110785256 申请日期 2011.11.09
申请人 BRISTOL-MYERS SQUIBB COMPANY 发明人 AUSTIN, JOEL F.;FRENNESSON, DAVID B.;SAULNIER, MARK G.
分类号 C07D471/04;A61K31/437;A61P35/00 主分类号 C07D471/04
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