发明名称 |
5-(ARYLSULFONYL)-PYRAZOLOPIPERIDINES |
摘要 |
THE INVENTION PROVIDES N-CYCLIC SULFONAMIDO COMPOUNDS OF FORMULA WHEREIN A, B, R?, R??, R?, R??, R? AND R?? ARE AS DESCRIBED IN THE SPECIFICATION. COMPOUNDS OF FORMULA I ARE USEFUL IN TREATING OR PREVENTING COGNITIVE DISORDERS, SUCH AS ALZHEIMER'S DISEASE. THE INVENTION ALSO ENCOMPASSES PHARMACEUTICAL COMPOSITIONS COMPRISING COMPOUNDS OF FORMULA I, METHODS OF PREPARING COMPOUNDS OF FORMULA I, AND METHODS OF TREATING COGNITIVE DISORDERS, SUCH AS ALZHEIMER'S DISEASE. |
申请公布号 |
MY149422(A) |
申请公布日期 |
2013.08.30 |
申请号 |
MY2008PI01060 |
申请日期 |
2006.12.01 |
申请人 |
ELAN PHARMACEUTICALS, INC. |
发明人 |
GAROFALO, ALBERT W.;JAGODZINSKI, JACEK J.;KONRADI, ANDREI W.;SEMKO, CHRISTOPHER M.;SMITH, JENIFER L.;XU, YING-ZI;YE, XIAOCONG MICHAEL |
分类号 |
C07D211/96 |
主分类号 |
C07D211/96 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|