发明名称 |
An improved process for preparation of levonorgestrel |
摘要 |
<p>The present invention provides an improved process for preparation of levonorgestrel (3) which comprises of hydrolysis of 13β-ethyl-3-methoxy-17α-ethynyl-gona-2,5(10)-dien-17β- o1 (2) with an acid in aprotic solvent. The present invention also provides a novel process for purification of crude levonorgestrel (3) by recrystallization from N,N-dimethyl formamide- water; methanol-water mixture.</p> |
申请公布号 |
AU2012219096(A1) |
申请公布日期 |
2013.08.29 |
申请号 |
AU20120219096 |
申请日期 |
2012.02.14 |
申请人 |
LUPIN LIMITED |
发明人 |
ZADBUKE, SWAPNIL AJIT;MEHARE, KISHOR GULABRAO;GODBOLE, HIMANSHU MADHAV;SINGH, GIRIJ PAL |
分类号 |
C07J1/00;C07J75/00 |
主分类号 |
C07J1/00 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|