发明名称 |
8 - SUBSTITUTED 2 -AMINO - [1,2,4] TRIAZOLO [1, 5 -A] PYRAZINES AS SYK TRYROSINE KINASE INHIBITORS AND GCN2 SERIN KINASE INHIBITORS |
摘要 |
Compounds of the formula I in which R1, R2 and R4 have the meanings indicated in Claim 1, are inhibitors of Syk, and can be employed, inter alia, for the treatment of cancer, rheumatoid arthritis and / or systemic lupus |
申请公布号 |
WO2013124026(A1) |
申请公布日期 |
2013.08.29 |
申请号 |
WO2013EP00189 |
申请日期 |
2013.01.22 |
申请人 |
MERCK PATENT GMBH |
发明人 |
DEUTSCH, CARL;KUHN, DANIEL;ROSS, TATJANA;BURGDORF, LARS |
分类号 |
C07D487/04;A61K31/4985;A61P25/00;A61P29/00;A61P35/00;C07D519/00 |
主分类号 |
C07D487/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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