发明名称 ONE POT PROCESS FOR PRODUCING 6-HYDROXYL NAL-OPIATE
摘要 The present invention provides processes for preparing nal-opiates without the isolation of intermediates. In general, the process provides for alkylation and reduction in the same pot to give the nal-opi- ate (I).
申请公布号 WO2013119886(A1) 申请公布日期 2013.08.15
申请号 WO2013US25244 申请日期 2013.02.08
申请人 MALLINCKRODT LLC 发明人 WANG, PETER, X.;JIANG, TAO;BERBERICH, DAVID, W.
分类号 C07D489/02;A61K31/485;C07D489/08 主分类号 C07D489/02
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