发明名称 |
ONE POT PROCESS FOR PRODUCING 6-HYDROXYL NAL-OPIATE |
摘要 |
The present invention provides processes for preparing nal-opiates without the isolation of intermediates. In general, the process provides for alkylation and reduction in the same pot to give the nal-opi- ate (I). |
申请公布号 |
WO2013119886(A1) |
申请公布日期 |
2013.08.15 |
申请号 |
WO2013US25244 |
申请日期 |
2013.02.08 |
申请人 |
MALLINCKRODT LLC |
发明人 |
WANG, PETER, X.;JIANG, TAO;BERBERICH, DAVID, W. |
分类号 |
C07D489/02;A61K31/485;C07D489/08 |
主分类号 |
C07D489/02 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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