发明名称 |
MORPHOLINO NUCLEIC ACID DERIVATIVE |
摘要 |
<p>The Present invention provides a useful morpholino nucleic acid derivative for synthesizing a morpholino nucleic acid oligomer.
The present invention provides a compound represented by the following general formula (1) or a salt.
wherein R 1 represents hydrogen, trityl and so on.
R 2 represents amide or imine.
R 3 represents a hydroxy group which may be protected by trialkylsilyl and so on, or a group represented by the following general formula (5).
(wherein X represents O or S. Y represents dialkylamino or alkoxy. Z represents chlorine.)</p> |
申请公布号 |
EP2623507(A1) |
申请公布日期 |
2013.08.07 |
申请号 |
EP20110829283 |
申请日期 |
2011.09.29 |
申请人 |
NIPPON SHINYAKU CO., LTD. |
发明人 |
UEDA, TOSHIHIRO |
分类号 |
C07F9/24;C07D473/18;C07F7/18;C07F9/6558;C07F9/6561 |
主分类号 |
C07F9/24 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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