发明名称 |
CYCLIC ENONE COMPOUND HAVING TDP1 INHIBITORY ACTIVITY |
摘要 |
<P>PROBLEM TO BE SOLVED: To provide a compound that has a strong Tyrosyl DNA Phosphodiesterase inhibitory activity, and can be used as pharmaceuticals. <P>SOLUTION: The cyclic enone compound is exemplified by formula (4f) and formula (4e), and a therapeutic agent of cancer and a method of a treatment of a cancer use the same. <P>COPYRIGHT: (C)2013,JPO&INPIT |
申请公布号 |
JP2013121930(A) |
申请公布日期 |
2013.06.20 |
申请号 |
JP20110270875 |
申请日期 |
2011.12.12 |
申请人 |
TOKYO INSTITUTE OF TECHNOLOGY;NATIONAL INSTITUTE OF ADVANCED INDUSTRIAL SCIENCE& TECHNOLOGY;JAPAN BIOLOGICAL INFORMATICS CONSORTIUM |
发明人 |
TAKAHASHI TAKASHI;DOI TAKAYUKI;FUSE SHINICHIRO;ARAYA KAZUO;TAKAGI MOTOKI;HIROKAWA TAKATSUGU;INABA KENICHI;TANAKA MASAHIRO |
分类号 |
C07D317/72;A61K31/357;A61K31/381;A61K31/443;A61K31/4709;A61K31/506;A61P35/00;A61P43/00;C07D405/10;C07D407/10;C07D409/10 |
主分类号 |
C07D317/72 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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