发明名称 4- { [ ( PYRIDIN- 3 - YL -METHYL) AMINOCARBONYL] AMINO} BENZENE - SULFONE DERIVATIVES AS NAMPT INHIBITORS FOR THERAPY OF DISEASES SUCH AS CANCER
摘要 <p>The present invention relates to compounds and compositions for the inhibition of NAMPT, their synthesis, applications and antidotes. An embodiment of the invention is the provision of a compound of Formula IIIA.</p>
申请公布号 WO2012031196(A9) 申请公布日期 2013.06.13
申请号 WO2011US50320 申请日期 2011.09.02
申请人 FORMA TM, LLC;GENENTECH, INC.;BAIR, KENNETH W.;BAUMEISTER, TIMM R.;BUCKMELTER, ALEXANDRE J.;CLODFELTER, KARL H.;HAN, BINGSONG;LIN, JIAN;REYNOLDS, DOMINIC J.;SMITH, CHASE C.;WANG, ZHONGGUO;ZHENG, XIAOZHANG;YUEN, PO-WAI 发明人 BAIR, KENNETH W.;BAUMEISTER, TIMM R.;BUCKMELTER, ALEXANDRE J.;CLODFELTER, KARL H.;HAN, BINGSONG;LIN, JIAN;REYNOLDS, DOMINIC J.;SMITH, CHASE C.;WANG, ZHONGGUO;ZHENG, XIAOZHANG;YUEN, PO-WAI
分类号 C07D213/54;A61K31/4406;A61K31/443;A61K31/4433;A61K31/4439;A61P35/00;C07C317/00;C07D213/74;C07D213/75;C07D213/81;C07D213/84;C07D471/04 主分类号 C07D213/54
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