| 发明名称 |
PREPARATION OF PROTECTED ALPHA-KETO BETA-AMINO ESTERS AND AMIDES |
| 摘要 |
The invention provides beta-sulfonamide alpha-keto esters and amides in which the alpha-keto is protected as a 1,3-dithiolane derivative. Also provided are methods for preparing such esters and amides and for incorporating them into peptides.
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| 申请公布号 |
US2013131356(A1) |
申请公布日期 |
2013.05.23 |
| 申请号 |
US201313735757 |
申请日期 |
2013.01.07 |
| 申请人 |
VERTEX PHAMACEUTICALS INCORPORATED;VERTEX PHAMACEUTICALS INCORPORATED |
发明人 |
NUGENT WILLIAM A.;LOOKER ADAM R.;FORSLUND RAYMOND E.;MARTINOT THEODORE A.;HARRISON CRISTIAN L.;IBRAHIM SHEREE |
| 分类号 |
C07D339/06 |
主分类号 |
C07D339/06 |
| 代理机构 |
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