发明名称 |
Azetidinyl diamides as monoacylglycerol lipase inhibitors |
摘要 |
Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula (I) as follows: wherein Y, Z, R1, and s are defined herein.
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申请公布号 |
US8445477(B2) |
申请公布日期 |
2013.05.21 |
申请号 |
US20100765048 |
申请日期 |
2010.04.22 |
申请人 |
BIAN HAIYAN;CHEVALIER KRISTEN;CLEMENTE JOSE;CONNOLLY PETE;FLORES CHRIS;LIN SHU-CHEN;LIU LI;MABUS JOHN;MACIELAG MARK;MCDONNELL MARK;PITIS PHILIP;ZHANG YUE-MEI;ZHANG SUI-PO;ZHU BIN;JANSSEN PHARMACEUTICA, NV |
发明人 |
BIAN HAIYAN;CHEVALIER KRISTEN;CLEMENTE JOSE;CONNOLLY PETE;FLORES CHRIS;LIN SHU-CHEN;LIU LI;MABUS JOHN;MACIELAG MARK;MCDONNELL MARK;PITIS PHILIP;ZHANG YUE-MEI;ZHANG SUI-PO;ZHU BIN |
分类号 |
A61K31/496;A61K31/541;A61K31/55;C07D205/04;C07D401/12;C07D403/04;C07D409/06;C07D413/12;C07D471/04;C07D491/048 |
主分类号 |
A61K31/496 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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