发明名称 Azetidinyl diamides as monoacylglycerol lipase inhibitors
摘要 Disclosed are compounds, compositions and methods for treating various diseases, syndromes, conditions and disorders, including pain. Such compounds are represented by Formula (I) as follows: wherein Y, Z, R1, and s are defined herein.
申请公布号 US8445477(B2) 申请公布日期 2013.05.21
申请号 US20100765048 申请日期 2010.04.22
申请人 BIAN HAIYAN;CHEVALIER KRISTEN;CLEMENTE JOSE;CONNOLLY PETE;FLORES CHRIS;LIN SHU-CHEN;LIU LI;MABUS JOHN;MACIELAG MARK;MCDONNELL MARK;PITIS PHILIP;ZHANG YUE-MEI;ZHANG SUI-PO;ZHU BIN;JANSSEN PHARMACEUTICA, NV 发明人 BIAN HAIYAN;CHEVALIER KRISTEN;CLEMENTE JOSE;CONNOLLY PETE;FLORES CHRIS;LIN SHU-CHEN;LIU LI;MABUS JOHN;MACIELAG MARK;MCDONNELL MARK;PITIS PHILIP;ZHANG YUE-MEI;ZHANG SUI-PO;ZHU BIN
分类号 A61K31/496;A61K31/541;A61K31/55;C07D205/04;C07D401/12;C07D403/04;C07D409/06;C07D413/12;C07D471/04;C07D491/048 主分类号 A61K31/496
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