发明名称 |
PREPARATION OF 13-CYCLOHEXYL-3-METHOXY-6-[METHYL-(2--ETHYL)-CARBAMOYL]-7H-INDOLO-[2,1-a]-[2]-BENZAZEPINE-10-CARBOXYLIC ACID |
摘要 |
The present invention relates to an improved method for the preparation of 13-cyclohexyl-3-methoxy-6-[methyl-(2-{2-[methyl-(sulphamoyl)-amino]-ethoxy}-ethyl)-carbamoyl]-7H-indolo-[2,1-a]-[2]-benzazepine-10-carboxylic acid. The present invention also relates to a new compound, namely tert-butyl (methyl-{2-[2-(methylamino)-ethoxy]-ethyl}-sulphamoyl)-carbamate, used in this improved method.
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申请公布号 |
US2013102777(A1) |
申请公布日期 |
2013.04.25 |
申请号 |
US201113805607 |
申请日期 |
2011.06.24 |
申请人 |
GOVAERTS TOM CORNELIS HORTENSE;BONGARTZ JEAN-PIERRE-ANDRE MARC;NIESTE PATRICK HUBERT J.;JANSSEN R&D IRELAND |
发明人 |
GOVAERTS TOM CORNELIS HORTENSE;BONGARTZ JEAN-PIERRE-ANDRE MARC;NIESTE PATRICK HUBERT J. |
分类号 |
C07D487/04;C07C307/06 |
主分类号 |
C07D487/04 |
代理机构 |
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地址 |
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