发明名称 PIPERIDINONE DERIVATIVES AS MDM2 INHIBITORS FOR THE TREATMENT OF CANCER
摘要 The present invention provides MDM2 inhibitor compounds of Formula IE, which compounds are useful as therapeutic agents, particularly for the treatment of cancers. The present invention also relates to pharmaceutical compositions that contain an MDM2 inhibitor.
申请公布号 EP2576510(A1) 申请公布日期 2013.04.10
申请号 EP20110726581 申请日期 2011.06.03
申请人 AMGEN INC. 发明人 BARTBERGER, MICHAEL DAVID;GONZALEZ BUENROSTRO, ANA;BECK, HILARY PLAKE;CHEN, XIAOQI;CONNORS, RICHARD VICTOR;DEIGNAN, JEFFREY;DUQUETTE, JASON;EKSTEROWICZ, JOHN;FISHER, BENJAMIN;FOX, BRIAN MATTHEW;FU, JIASHENG;FU, ZICE;GONZALEZ LOPEZ DE TURISO, FELIX;GRIBBLE, JR., MICHAEL WILLIAM;GUSTIN, DARIN JAMES;HEATH, JULIE ANNE;HUANG, XIN;JIAO, XIANYUN;JOHNSON, MICHAEL;KAYSER, FRANK;KOPECKY, DAVID JOHN;LAI, SUJEN;LI, YIHONG;LI, ZHIHONG;LIU, JIWEN;LOW, JONATHAN DANTE;LUCAS, BRIAN STUART;MA, ZHIHUA;MCGEE, LAWRENCE;MCINTOSH, JOEL;MCMINN, DUSTIN;MEDINA, JULIO CESAR;MIHALIC, JEFFREY THOMAS;OLSON, STEVEN HOWARD;REW, YOSUP;ROVETO, PHILIP MARLEY;SUN, DAQING;WANG, XIAODONG;WANG, YINGCAI;YAN, XUELEI;YU, MING;ZHU, JIANG
分类号 C07D211/40;A61K31/4412;A61P35/00;C07D279/02;C07D401/04;C07D401/06;C07D401/12;C07D407/04;C07D407/06;C07D409/04;C07D413/06;C07D417/06;C07D471/20;C07D498/08;C07D498/20 主分类号 C07D211/40
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