发明名称 ESTRA-1,3,5(10),16-TETRAENE-3-CARBOXAMIDE DERIVATIVES, PROCESS FOR PREPARATION THEREOF, PHARMACEUTICAL PREPARATIONS COMPRISING THEM, AND USE THEREOF FOR PRODUCTION OF MEDICAMENTS
摘要 The invention relates to AKR1C3 inhibitors and to processes for preparation thereof, to the use thereof for treatment and/or prophylaxis of diseases and to the use thereof for production of medicaments for treatment and/or prophylaxis of diseases, especially of bleeding problems and endometriosis.
申请公布号 WO2013045407(A1) 申请公布日期 2013.04.04
申请号 WO2012EP68803 申请日期 2012.09.24
申请人 BAYER INTELLECTUAL PROPERTY GMBH;BAYER PHARMA AKTIENGESELLSCHAFT 发明人 BOTHE, ULRICH;BARAK, NAOMI;BUSEMANN, MATTHIAS;FISCHER, OLIVER MARTIN;ROTGERI, ANDREA;GASHAW, ISABELLA;HARTUNG, INGO;MARQUARDT, TOBIAS
分类号 C07J43/00;A61K31/58;A61P5/24 主分类号 C07J43/00
代理机构 代理人
主权项
地址