发明名称 CYCLOALKYLNITRILE PYRAZOLE CARBOXAMIDES AS JANUS KINASE INHIBITORS
摘要 Cycloalkylnitrile pyrazole carboxamides as JAK inhibitors useful for the treatment of JAK-mediated diseases such as rheumatoid arthritis, asthma, COPD and cancer are provided.
申请公布号 WO2013040863(A1) 申请公布日期 2013.03.28
申请号 WO2012CN01291 申请日期 2012.09.21
申请人 MERCK SHARP & DOHME CORP.;BRUBAKER, JASON;DINSMORE, CHRISTOPHER J.;HOFFMAN, DAWN MARIE;JUNG, JOON;LIU, DUAN;PETERSON, SCOTT;SIU, TONY;TORRES, LUIS E.;ZHANG, HONGJUN;WEI, ZHONGYONG;SHI, FENG 发明人 BRUBAKER, JASON;DINSMORE, CHRISTOPHER J.;HOFFMAN, DAWN MARIE;JUNG, JOON;LIU, DUAN;PETERSON, SCOTT;SIU, TONY;TORRES, LUIS E.;ZHANG, HONGJUN;WEI, ZHONGYONG;SHI, FENG
分类号 C07D231/10;A61K31/415;A61P35/00;A61P37/00 主分类号 C07D231/10
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