发明名称 |
Indole derivatives as CRTH2 receptor antagonists |
摘要 |
Compound of formula I are antagonists of the PGD2 receptor, CRTH2, and as such are useful in the treatment and/or prevention of CRTH2-mediated diseases such as asthma.
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申请公布号 |
US8394819(B2) |
申请公布日期 |
2013.03.12 |
申请号 |
US20100708924 |
申请日期 |
2010.02.19 |
申请人 |
BERTHELETTE CARL;BOYD MICHAEL;COLUCCI JOHN;VILLENEUVE KARINE;METHOT JOEY;MERCK SHARP & DOHME CORP. |
发明人 |
BERTHELETTE CARL;BOYD MICHAEL;COLUCCI JOHN;VILLENEUVE KARINE;METHOT JOEY |
分类号 |
A61K31/404;A61K31/4353;C07D451/02;C07D487/04 |
主分类号 |
A61K31/404 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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