| 发明名称 |
METHOD FOR MONOFLUOROMETHYLATION OF ORGANIC SUBSTRATES TO PREPARE BIOLOGICALLY ACTIVE ORGANIC COMPOUNDS |
| 摘要 |
<p>The present invention describes a process for the preparation of monofluoromethylated organic biologically active compounds using monofluoromethylated reagents. Fluticasone Propionate and Fluticasone Furoate can be prepared using, for example, S-monofluoromethyl-S-phenyl-2,3,4,5- tetramethylphenylsulfonium tetrafluoroborate as monofluoromethylating reagent instead of bromofluoromethane.</p> |
| 申请公布号 |
WO2011151624(A8) |
申请公布日期 |
2013.03.07 |
| 申请号 |
WO2011GB00834 |
申请日期 |
2011.06.01 |
| 申请人 |
HOVIONE INTER LIMITED;LEITAO, EMILIA PERPETUA TAVARES;TURNER, CRAIG ROBERT |
发明人 |
LEITAO, EMILIA PERPETUA TAVARES |
| 分类号 |
C07J31/00 |
主分类号 |
C07J31/00 |
| 代理机构 |
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