发明名称 |
PROCESS FOR THE PREPARATION OF EPOXIDES AS INTERMEDIATES FOR THE SYNTHESIS OF NEBIVOLOL |
摘要 |
<p>The present invention relates to a novel process of synthesis of epoxides, 6-fluoro-2- (oxiran-2-yl) chroman (Figure 1), intermediates for the synthesis of nebivolol, depicted in Scheme (1), enabling to obtain the above- mentioned epoxides in a racemic or semichiral form.</p> |
申请公布号 |
WO2013018053(A1) |
申请公布日期 |
2013.02.07 |
申请号 |
WO2012IB53956 |
申请日期 |
2012.08.02 |
申请人 |
MENARINI INTERNATIONAL OPERATIONS LUXEMBOURG S.A.;CIPOLLONE, AMALIA;D'ANDREA, PIERO;FATTORI, DANIELA |
发明人 |
CIPOLLONE, AMALIA;D'ANDREA, PIERO;FATTORI, DANIELA |
分类号 |
C07D311/58;C07D407/04 |
主分类号 |
C07D311/58 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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