发明名称 CRYSTAL OF DIAMINE DERIVATIVE AND METHOD OF PRODUCING SAME
摘要 An object of the present invention is to provide a novel crystal form of a compound that has an inhibitory effect on activated blood coagulation factor X and is useful as a pharmaceutical compound for prevention and/or treatment of thrombotic and/or embolic diseases. The present invention provides a novel crystal form of N1-(5-chloropyridin-2-yl)-N2-((1S,2R,4S)-4-[(dimethylamino)carbonyl]-2-{[(5-methyl-4,5,6,7-tetrahydrothiazolo[5,4-c]pyridin-2-yl)carbonyl]amino}cyclohexyl)ethanediamide p-toluenesulfonate monohydrate, and method for producing the same.
申请公布号 US2013035356(A1) 申请公布日期 2013.02.07
申请号 US201213622783 申请日期 2012.09.19
申请人 DAIICHI SANKYO COMPANY, LIMITED;DAIICHI SANKYO COMPANY, LIMITED 发明人 SUZUKI TETSUYA;ONO MAKOTO
分类号 C07D513/04;A61K31/444;A61P7/02;A61P9/10 主分类号 C07D513/04
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