发明名称 |
NOVEL MODULATORS OF SPHINGOSINE PHOSPHATE RECEPTORS |
摘要 |
Compounds that activate a sphingosine-1-phosphate receptor of the subtype 1 are provided. Certain compounds selectively activate the receptor subtype 1 in relation to the sphinogosine-1-phosphate receptor subtype 3. Uses and methods of inventive compounds for treatment of malconditions wherein activation, agonism, inhibition or antagonism of the S1P1 is medically indicated are provided. |
申请公布号 |
US2012329840(A1) |
申请公布日期 |
2012.12.27 |
申请号 |
US201213605561 |
申请日期 |
2012.09.06 |
申请人 |
ROBERTS EDWARD;ROSE HUGH;BROWN STEVEN;GUERRERO MIGUEL A.;PENG XUEMEI;PODDUTOORI RAMULU;THE SCRIPPS RESEARCH INSTITUTE |
发明人 |
ROBERTS EDWARD;ROSE HUGH;BROWN STEVEN;GUERRERO MIGUEL A.;PENG XUEMEI;PODDUTOORI RAMULU |
分类号 |
A61K31/4245;A61P11/00;A61P25/00;A61P37/06;C07D271/06 |
主分类号 |
A61K31/4245 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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