发明名称 AMINO-TETRAZOLES ANALOGUES AND METHODS OF USE
摘要 A compound having Formula (I) or Formula (II) is disclosed as an P2X7 antagonist, wherein A, B, C, Y, Y, Z, m, v, R1, R2, R3, R4, and R5, are as defined in the description. Methods and compositions for treating disease or condition modulated by P2X7 are also disclosed.
申请公布号 US2012329772(A1) 申请公布日期 2012.12.27
申请号 US201213544387 申请日期 2012.07.09
申请人 CARROLL WILLIAM A.;PEREZ-MEDRANO ARTURO;FLORJANCIC ALAN S.;NELSON DEREK W.;PEDDI SRIDHAR;LI TONGMEI;BUNNELLE ERIC M.;HIRST GAVIN;LI BIQIN C.;ABBOTT LABORATORIES 发明人 CARROLL WILLIAM A.;PEREZ-MEDRANO ARTURO;FLORJANCIC ALAN S.;NELSON DEREK W.;PEDDI SRIDHAR;LI TONGMEI;BUNNELLE ERIC M.;HIRST GAVIN;LI BIQIN C.
分类号 C07D257/06;A61K31/41;A61K31/4155;A61K31/427;A61K31/435;A61K31/4355;A61K31/4439;A61K31/444;A61K31/4709;A61K31/496;A61K31/497;A61K31/506;A61K31/5377;A61K31/55;A61K31/551;A61K31/553;A61P25/00;A61P25/24;A61P25/28;A61P29/00;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D405/12;C07D409/12;C07D409/14;C07D413/12;C07D413/14;C07D417/12;C07D417/14;C07D487/04;C07D491/04;C07D491/048;C07D491/18 主分类号 C07D257/06
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