发明名称 |
AKT / PKB INHIBITORS |
摘要 |
The invention relates to a series of compounds with particular activity as inhibitors of the serine-threonine kinase AKT. Also provided are pharmaceutical compositions comprising same as well as methods for treating cancer.
|
申请公布号 |
US2012309739(A1) |
申请公布日期 |
2012.12.06 |
申请号 |
US201013508137 |
申请日期 |
2010.11.03 |
申请人 |
BELL MARK PETER;O'DOWD COLIN RODERICK;ROUNTREE JAMES SAMUEL SHANE;TREVITT GRAHAM PETER;HARRISON TIMOTHY;MCFARLAND MARY MELISSA;ALMAC DISCOVERY LIMITED |
发明人 |
BELL MARK PETER;O'DOWD COLIN RODERICK;ROUNTREE JAMES SAMUEL SHANE;TREVITT GRAHAM PETER;HARRISON TIMOTHY;MCFARLAND MARY MELISSA |
分类号 |
A61K31/4355;A61K31/343;A61K31/353;A61K31/397;A61K31/4985;A61K31/519;A61K31/5377;A61P35/00;C07D307/81;C07D311/36;C07D405/10;C07D491/048 |
主分类号 |
A61K31/4355 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|