4H-THIENO[3,2-C]CHROMENE-BASED INHIBITORS OF NOTUM PECTINACETYLESTERASE AND METHODS OF THEIR USE
摘要
Compounds that may be used to inhibit Notum Pectinacetylesterase are described, as well as compositions comprising them, and methods of their use to treat diseases and disorders affecting bone.
申请公布号
CA2837084(A1)
申请公布日期
2012.12.06
申请号
CA20122837084
申请日期
2012.05.23
申请人
LEXICON PHARMACEUTICALS, INC.
发明人
BARBOSA, JOSEPH;CARSON, KENNETH GORDON;GARDYAN, MICHAEL WALTER;HEALY, JASON PATRICK;HAN, QIANG;MABON, ROSS;PRAVEEN, PABBA;TARVER, JAMES, JR.;TERRANOVA, KRISTEN M.;TUNOORI, ASHOK;XU, XIAOLIAN