发明名称 PROCESS FOR RILPIVIRINE
摘要 <p>The present invention provides a novel process for the preparation of 4-(4-hydroxypyrimidin-2-ylamino)benzonitrile. The present invention also provides a novel process for the preparation of 4-iodo-2,6-dimethyl benzenamine. The present invention further provides an improved process for the preparation of rilpivirine. The present invention further provides a tosylate salt of rilpivirine, process for its preparation and pharmaceutical compositions comprising it.</p>
申请公布号 CA2834257(A1) 申请公布日期 2012.11.01
申请号 CA20122834257 申请日期 2012.02.16
申请人 HETERO RESEARCH FOUNDATION 发明人 PARTHASARADHI REDDY, BANDI;RATHNAKAR REDDY, KURA;MURALIDHARA REDDY, DASARI;VENKAT NARSIMHA REDDY, ADULLA;VAMSI KRISHNA, BANDI
分类号 C07D239/47 主分类号 C07D239/47
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