发明名称 Age Inhibitors
摘要 The invention relates to a compound having general formula I, wherein: X represents CH2, C═O, C═S or CHOH, R1 represents an amino acid optionally substituted by one or more halogen atoms, or by one or more CF3 groups and n=0.1 or 2, or R1 represents a peptide containing two amino acids, each amino acid being optionally substituted by one or more halogen atoms, or by one or more CF3 groups and n=0 or 1, or XR1 represent PO3H or SO3H and n=0.1 or 2; R2 represents H, XR1, an alkyl group at C1-C6, an aralkyl group at C1-C6 or an aryl group, whereby the alkyl, aralkyl and aryl groups can be substituted by an amine NH2, a carboxylic group COOH, one or more halogen atoms.
申请公布号 US2012252866(A1) 申请公布日期 2012.10.04
申请号 US201213437491 申请日期 2012.04.02
申请人 POTIER PIERRE;POTIER GUY JEAN MARIE;ZELVEYAN MARIE CLAUDE DENISE MICHELE;MAGNAN CATHERINE MARIE GERMAINE;DRION ODETTE;SASAKI NOBUMICHI ANDRE;ACHAB GARCIA ALVAREZ MARIA CONCEPCION;WANG-ZHU QIAN;ERMOLENKO LIOUDMILA;BAKALA JOANNA;FRANCK GISELE;BAKRIM NHIRI NAIMA;CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS);PHARMAMENS 发明人 POTIER PIERRE;POTIER GUY JEAN MARIE;ZELVEYAN MARIE CLAUDE DENISE MICHELE;MAGNAN CATHERINE MARIE GERMAINE;DRION ODETTE;SASAKI NOBUMICHI ANDRE;ACHAB GARCIA ALVAREZ MARIA CONCEPCION;WANG-ZHU QIAN;ERMOLENKO LIOUDMILA;BAKALA JOANNA;FRANCK GISELE;BAKRIM NHIRI NAIMA
分类号 A61K8/36;A61K8/37;A61K8/49;A61Q19/08 主分类号 A61K8/36
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