发明名称 |
1,3,4,8-TETRAHYDRO-2H-PYRIDO[1,2-A]PYRAZINE DERIVATIVE AND USE OF SAME AS HIV INTEGRASE INHIBITOR |
摘要 |
<p>•1,3,4,8-TETRAHYDRO-2H-PYRIDO11,2-AlPYRAZINE DERIVATIVE AND USE OF SAME AS HIV INTEGRASE INHIBITORProvided is a nuVe1•1,3,4,8-tetrahydro-2H-pyrido[1,2- a]pyrazine derivative or a pharmaceutically acceptable salt5 thereof, or a solvate thereof, which is useful as an anti-HIV agent.The present invention provides a compound represented by the following formula [I]OH 0 / 1 5y----N10 wherein each symbol is as defined in the specification, or a pharmaceutically acceptable salt thereof, or a solvate thereof.</p> |
申请公布号 |
SG183484(A1) |
申请公布日期 |
2012.09.27 |
申请号 |
SG20120062881 |
申请日期 |
2011.02.25 |
申请人 |
JAPAN TOBACCO INC. |
发明人 |
MIYAZAKI, SUSUMU;BESSHO, YUKI;ADACHI, KAORU;KAWASHITA, SEIJI;ISOSHIMA, HIROTAKA;OSHITA, KENGO;FUKUDA, SHUNICHI |
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