发明名称 Polymorph B of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a]pyrimidin-7-yl]-phenyl}-N-methyl-acetamide
摘要 The present invention relates to a method of treating anxiety, epilepsy, sleep disorders, and insomnia, for inducing sedation-hypnosis, anesthesia, and muscle relaxation, and for modulating the necessary time to induce sleep and its duration, which comprises administering a therapeutically effective amount of Polymorph B of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a]pyrimidin-7-yl]-phenyl}-N-methyl-acetamide characterized by a powder X-Ray diffraction pattern containing specific peaks at 2&thetas;=7.1° (±0.1°) and 21.4° (±0.1°) to a patient in need thereof.
申请公布号 US8273753(B2) 申请公布日期 2012.09.25
申请号 US201113115272 申请日期 2011.05.25
申请人 ANGLADA LUIS;PALOMER ALBERT;GUGLIETTA ANTONIO;FERRER INTERNATIONAL, S.A. 发明人 ANGLADA LUIS;PALOMER ALBERT;GUGLIETTA ANTONIO
分类号 A01N43/90;A61K31/519;C07D487/00 主分类号 A01N43/90
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