发明名称 |
SYNTHETIC INTERMEDIATE OF OXAZOLE COMPOUND AND METHOD FOR PRODUCING THE SAME. |
摘要 |
<p>An object of the present invention is to provide a method for producing an oxazole compound in a high yield. The object can be achieved by a compound represented by Formula (11): wherein R1 is a hydrogen atom or lower-alkyl group; R2 is a 1-piperidyl group substituted at the 4-position with a substituent selected from (A1a) a phenoxy group substituted on the phenyl moiety with one or more halogen-substituted lower-alkoxy groups, (A1b) a phenoxy-substituted lower-alkyl group substituted on the phenyl moiety with one or more halogen-substituted lower-alkyl groups, (A1c) a phenyl-substituted lower-alkoxy lower-alkyl group substituted on the phenyl moiety with halogen, (A1d) a phenyl-substituted lower-alkyl group substituted on the phenyl moiety with one or more halogen-substituted lower-alkoxy groups, (A1e) an amino group substituted with a phenyl group substituted with one or more halogen-substituted lower-alkoxy groups, and a lower-alkyl group, and (A1f) a phenyl-substituted lower-alkoxy group substituted on the phenyl moiety with one or more halogen-substituted lower-alkoxy groups; n is an integer from 1 to 6; and X3 is an organic sulfonyloxy group.</p> |
申请公布号 |
MX2012008501(A) |
申请公布日期 |
2012.08.17 |
申请号 |
MX20120008501 |
申请日期 |
2011.01.28 |
申请人 |
OTSUKA PHARMACEUTICAL CO., LTD.* |
发明人 |
SHINHAMA, KOICHI;UTSUMI, NAOTO;AKI, SHINJI;FUJITA, NOBUHISA;YAMAMOTO, AKIHIRO;OGASAWARA, SHIN |
分类号 |
C07D211/46;C07D405/12;C07D498/04 |
主分类号 |
C07D211/46 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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