发明名称 |
Derivatives of pyrimido[6,1-A]isoquinolin-4-one |
摘要 |
The present invention relates to derivatives of pyrimido[6,1-a]isoquinolin-4-one and their application as inhibitors of phosphodiesterase (PDE) isoenzymes. More particularly the invention relates to derivatives of pyrimido[6,1-a]isoquinolin-4-one and their use in medicine for example as bronchodilators with anti-inflammatory properties. |
申请公布号 |
US8242127(B2) |
申请公布日期 |
2012.08.14 |
申请号 |
US20080150232 |
申请日期 |
2008.04.24 |
申请人 |
OXFORD ALEXANDER WILLIAM;JACK DAVID;VERONA PHARMA PLC |
发明人 |
OXFORD ALEXANDER WILLIAM;JACK DAVID |
分类号 |
A01N43/54;A61K9/12;A61K31/505;A61K31/519;A61P11/00;A61P11/06;A61P11/08;A61P43/00;C07D471/04 |
主分类号 |
A01N43/54 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|