发明名称 |
Substituted imidazopyridine derivatives as melanocortin-4 receptor antagonists |
摘要 |
The present invention relates to substituted imidazopyridine derivatives as melanocortin-4 receptor (MC-4R) modulators, in particular as melanocortin-4 receptor antagonists. The antagonists are useful for the treatment of disorders and diseases such as cancer cachexia, muscle wasting, anorexia, amytrophic lateral sclerosis (ALS), anxiety and depression. |
申请公布号 |
US8236818(B2) |
申请公布日期 |
2012.08.07 |
申请号 |
US20080530676 |
申请日期 |
2008.03.28 |
申请人 |
METZ GUENTHER;DEPPE HOLGER;ABEL ULRICH;FEURER ACHIM;OTT INGE;NORDHOFF SONJA;SOEBERDT MICHAEL;HOFFMANN-ENGER BARBARA;WEYERMANN PHILIPP;SIENDT HERVE;RUMMEY CHRISTIAN;TERINEK MIROSLAV;HENNEBOEHLE MARCO;HERZNER HOLGER;MONDADORI CESARE;SANTHERA PHARMACEUTICALS (SCHWEIZ) AG |
发明人 |
METZ GUENTHER;DEPPE HOLGER;ABEL ULRICH;FEURER ACHIM;OTT INGE;NORDHOFF SONJA;SOEBERDT MICHAEL;HOFFMANN-ENGER BARBARA;WEYERMANN PHILIPP;SIENDT HERVE;RUMMEY CHRISTIAN;TERINEK MIROSLAV;HENNEBOEHLE MARCO;HERZNER HOLGER;MONDADORI CESARE |
分类号 |
A61K31/437;C07D471/04 |
主分类号 |
A61K31/437 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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