发明名称 Tricyclic pyrazolopyrimidine derivatives
摘要 A pyrazolopyrimidine compound represented by formula (1) that inhibits the function of HSP90 as a chaperone protein and that has antitumor activity, a medicament comprising a compound represented by formula (1), a pharmaceutical composition comprising a compound represented by formula (1), and a method for treating cancer using a compound represented by formula (1).
申请公布号 US8236813(B2) 申请公布日期 2012.08.07
申请号 US20100915982 申请日期 2010.10.29
申请人 OHKI HITOSHI;OKAYAMA TOORU;IKEDA MASAHIRO;OTA MASAHIRO;SHIBATA YOSHIHIRO;NAKANISHI TOSHIYUKI;UEDA YASUSI;SUZUKI NOBUYUKI;MATUURA SHINJI;DAIICHI SANKYO COMPANY, LIMITED 发明人 OHKI HITOSHI;OKAYAMA TOORU;IKEDA MASAHIRO;OTA MASAHIRO;SHIBATA YOSHIHIRO;NAKANISHI TOSHIYUKI;UEDA YASUSI;SUZUKI NOBUYUKI;MATUURA SHINJI
分类号 C07D491/00;A01N43/54;A61K31/505;C07D239/00;C07D471/00;C07D487/00 主分类号 C07D491/00
代理机构 代理人
主权项
地址