发明名称 |
Tricyclic pyrazolopyrimidine derivatives |
摘要 |
A pyrazolopyrimidine compound represented by formula (1) that inhibits the function of HSP90 as a chaperone protein and that has antitumor activity, a medicament comprising a compound represented by formula (1), a pharmaceutical composition comprising a compound represented by formula (1), and a method for treating cancer using a compound represented by formula (1). |
申请公布号 |
US8236813(B2) |
申请公布日期 |
2012.08.07 |
申请号 |
US20100915982 |
申请日期 |
2010.10.29 |
申请人 |
OHKI HITOSHI;OKAYAMA TOORU;IKEDA MASAHIRO;OTA MASAHIRO;SHIBATA YOSHIHIRO;NAKANISHI TOSHIYUKI;UEDA YASUSI;SUZUKI NOBUYUKI;MATUURA SHINJI;DAIICHI SANKYO COMPANY, LIMITED |
发明人 |
OHKI HITOSHI;OKAYAMA TOORU;IKEDA MASAHIRO;OTA MASAHIRO;SHIBATA YOSHIHIRO;NAKANISHI TOSHIYUKI;UEDA YASUSI;SUZUKI NOBUYUKI;MATUURA SHINJI |
分类号 |
C07D491/00;A01N43/54;A61K31/505;C07D239/00;C07D471/00;C07D487/00 |
主分类号 |
C07D491/00 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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