发明名称 RING-FUSED COMPOUND
摘要 The present invention relates to: a compound having a URAT1 inhibitory activity; and an URAT1 inhibitor, a blood uric acid level reducing agent and a pharmaceutical composition, each of which comprises the compound. More specifically, the present invention relates to a compound represented by formula (I). [In the formula, R1 represents -Q1-A1 or the like; AA represents a double bond or a single bond; W1 represents a nitrogen atom or a group represented by general formula: =C(Ra)- and W2 represents a nitrogen atom or a group represented by general formula: =C(Rb)- when AA represents a double bond; W1 represents a group represented by general formula: -C(Raa)(Rab)- or a group represented by general formula: -(C=O)- and W2 represents a group represented by general formula: -C(Rba)(Rbb)-, a group represented by general formula: -(C=O)- or a group represented by general formula: -N(Rbc)- when AA represents a single bond; W3, W4 and W5 independently represent a nitrogen atom, a methine group which may have a substituentor the like; X represents a single bond, an oxygen atom or the like; Y represents a single bond or (CRYiRYi')n; and Z represents a hydroxy group, COOR2 or the like.]
申请公布号 WO2012102405(A1) 申请公布日期 2012.08.02
申请号 WO2012JP52009 申请日期 2012.01.30
申请人 SATO PHARMACEUTICAL CO., LTD.;NAGAI KEITA;NAGASAWA KOH;TAKAHASHI HIROBUMI;BABA MOTOAKI;FUJIOKA SHINICHI;KONDOH ERI;TANAKA KENICHI;ITOH YOSHIKI 发明人 NAGAI KEITA;NAGASAWA KOH;TAKAHASHI HIROBUMI;BABA MOTOAKI;FUJIOKA SHINICHI;KONDOH ERI;TANAKA KENICHI;ITOH YOSHIKI
分类号 C07D209/08;A61K31/404;A61K31/416;A61K31/4184;A61K31/4439;A61P9/10;A61P13/04;A61P13/12;A61P19/02;A61P19/06;A61P43/00;C07D209/30;C07D231/56;C07D235/08;C07D235/10;C07D401/06;C07D405/06 主分类号 C07D209/08
代理机构 代理人
主权项
地址