发明名称 |
APPLICATION OF TRIINDOLYL METHANE DERIVATIVES AS ANTICANCER DRUGS |
摘要 |
FIELD: medicine, pharmaceutics. ^ SUBSTANCE: invention refers to pharmaceutics and medicine and concerns triindolyl methane derivatives of formula ^ and as anticancer drugs showing cytotoxic, apoptotic action on tumour cells, and also blocking NFkB transcription factor activity. ^ EFFECT: compounds exhibit high anticancer activity. ^ 4 dwg, 3 tbl, 4 ex |
申请公布号 |
RU2454232(C2) |
申请公布日期 |
2012.06.27 |
申请号 |
RU20100138202 |
申请日期 |
2010.09.16 |
申请人 |
FEDERAL'NOE GOSUDARSTVENNOE BJUDZHETNOE UCHREZHDENIE "ROSSIJSKIJ ONKOLOGICHESKIJ NAUCHNYJ TSENTR IMENI N.N. BLOKHINA" ROSSIJSKOJ AKADEMII MEDITSINSKIKH NAUK (FGBU "RONTS IM. N.N. BLOKHINA" RAMN);UCHREZHDENIE ROSSIJSKOJ AKADEMII MEDITSINSKIKH NAUK NAUCHNO-ISSLEDOVATEL'SKIJ INSTITUT PO IZYSKANIJU NOVYKH ANTIBIOTIKOV IM. G.F. GAUZE RAMN (NIINA IM. G.F. GAUZE RAMN);ROSSIJSKAJA FEDERATSIJA V LITSE MINISTERSTVA OBRAZOVANIJA I NAUKI ROSSIJSKOJ FEDERATSII |
发明人 |
LAVRENOV SERGEJ NIKOLAEVICH;ISAKOVA ELENA BORISOVNA;PREOBRAZHENSKAJA MARIJA NIKOLAEVNA;TRESHCHALIN IVAN DMITRIEVICH;LICHINITSER MIKHAIL ROMANOVICH;STEPANOVA EVGENIJA VLADISLAVOVNA;SOLOMKO EHLISO SHALIKOVNA;ABRAMOV MIKHAIL EVGEN'EVICH;SHTIL' ALEKSANDR AL'BERTOVICH;BUKHMAN VLADIMIR MIKHAJLOVICH |
分类号 |
A61K31/404;A61P35/00 |
主分类号 |
A61K31/404 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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