发明名称 PROCESS FOR PREPARING A CHIRAL INTERMEDIATE FOR THE PREPARTION OF PITAVASTATIN
摘要 PURPOSE: A method for preparing chiral intermediates for producing pitavastatin is provided to simply obtain the chiral intermediates of high yield and high optical purity. CONSTITUTION: A method for preparing diol compound of chemical formula I comprises: a step of performing addition reaction of a compound of chemical formula II with a compound of chemical formula A to prepare a compound of chemical formula III; a step of deprotecting the compound of chemical formula III to prepare a compound of chemical formula IV; and a step of stereoselectively reducing the compound of chemical formula IV.
申请公布号 KR20120059148(A) 申请公布日期 2012.06.08
申请号 KR20100120782 申请日期 2010.11.30
申请人 CLS LABORATORIES, INC. 发明人 LIM, KWANG MIN
分类号 C07D215/04;C07D215/12 主分类号 C07D215/04
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