发明名称 LOW HYGROSCOPIC ARIPIPRAZOLE DRUG SUBSTANCE AND PROCESSES FOR THE PREPARATION THEREOF
摘要 The present invention provides low hygroscopic forms of aripiprazole and processes for the preparation thereof which will not convert to a hydrate or lose their original solubility even when a medicinal preparation containing the aripiprazole anhydride crystals is stored for an extended period.
申请公布号 HK1129891(A1) 申请公布日期 2012.06.08
申请号 HK20090107690 申请日期 2009.08.21
申请人 OTSUKA PHARMACEUTICAL CO. LTD. 发明人 TAKUJI BANDO;SATOSHI AOKI;JUNICHI KAWASAKI;MAKOTO ISHIGAMI;YOUICHI TANIGUCHI;TSUYOSHI YABUUCHI;KIYOSHI FUJIMOTO;YOSHIHIRO NISHIOKA;NORIYUKI KOBAYASHI;TSUTOMU FUJIMURA;MASANORI TAKAHASHI;KAORU ABE;TOMONORI NAKAGAWA;KOICHI SHINHAMA;NAOTO UTSUMI;MICHIAKI TOMINAGA;YOSHIHIRO OI;SHOHEI YAMADA;KENJI TOMIKAWA
分类号 C07D215/22;A61K;A61K9/14;A61K9/16;A61K9/20;A61K31/4704;A61K31/496;A61K31/501;A61P;A61P1/08;A61P3/04;A61P15/10;A61P25/00;A61P25/04;A61P25/16;A61P25/18;A61P25/22;A61P25/28;A61P25/32;B01D9/02;C07D;C07D215/227 主分类号 C07D215/22
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