发明名称 |
LOW HYGROSCOPIC ARIPIPRAZOLE DRUG SUBSTANCE AND PROCESSES FOR THE PREPARATION THEREOF |
摘要 |
The present invention provides low hygroscopic forms of aripiprazole and processes for the preparation thereof which will not convert to a hydrate or lose their original solubility even when a medicinal preparation containing the aripiprazole anhydride crystals is stored for an extended period. |
申请公布号 |
HK1129891(A1) |
申请公布日期 |
2012.06.08 |
申请号 |
HK20090107690 |
申请日期 |
2009.08.21 |
申请人 |
OTSUKA PHARMACEUTICAL CO. LTD. |
发明人 |
TAKUJI BANDO;SATOSHI AOKI;JUNICHI KAWASAKI;MAKOTO ISHIGAMI;YOUICHI TANIGUCHI;TSUYOSHI YABUUCHI;KIYOSHI FUJIMOTO;YOSHIHIRO NISHIOKA;NORIYUKI KOBAYASHI;TSUTOMU FUJIMURA;MASANORI TAKAHASHI;KAORU ABE;TOMONORI NAKAGAWA;KOICHI SHINHAMA;NAOTO UTSUMI;MICHIAKI TOMINAGA;YOSHIHIRO OI;SHOHEI YAMADA;KENJI TOMIKAWA |
分类号 |
C07D215/22;A61K;A61K9/14;A61K9/16;A61K9/20;A61K31/4704;A61K31/496;A61K31/501;A61P;A61P1/08;A61P3/04;A61P15/10;A61P25/00;A61P25/04;A61P25/16;A61P25/18;A61P25/22;A61P25/28;A61P25/32;B01D9/02;C07D;C07D215/227 |
主分类号 |
C07D215/22 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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