| 发明名称 |
Process for the preparation of fosinopril and intermediates thereof |
| 摘要 |
The present invention relates to a process for the preparation of intermediates useful in the synthesis of [1[S(R)],2±,4²]-4-cyclohexyl-1-[[[2-methyl-1-oxypropoxy) propoxy](4-phenylbutyl phosphinyl]acetyl]-L-proline, and the synthesis thereof, in particular as sodium salt (fosinopril sodium).
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| 申请公布号 |
EP2460808(A1) |
申请公布日期 |
2012.06.06 |
| 申请号 |
EP20110190979 |
申请日期 |
2011.11.28 |
| 申请人 |
DIPHARMA FRANCIS S.R.L. |
发明人 |
ALLEGRINI, PIETRO;ATTOLINO, EMANUELE;DE MARCO, ALESSANDRO;GORASSINI, FAUSTO;MICHIELETTI, MARIO |
| 分类号 |
C07F9/32 |
主分类号 |
C07F9/32 |
| 代理机构 |
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