发明名称 METHOD FOR PREPARING 5-CHLORO-N-(METHYL)THIOPHEN-2-CARBOXAMIDE DERIVATIVE AND INTERMEDIATE USED THEREIN
摘要 Disclosed are: a method for preparing a 5-chloro-N-({(5S)-2-oxo-3-[4-(5,6-dihydro-4H-[1,2,4]triazin-1-yl)phenyl]-1,3-oxazolidin-5-yl}-methyl)thiophene-2-carboxamide derivative, which is a inhibitor of blood coagulation factor Xa, in a high purity and yield; and a novel intermedicate used therein.
申请公布号 US2012136149(A1) 申请公布日期 2012.05.31
申请号 US201013382235 申请日期 2010.07.07
申请人 CHO YOUNG LAG;CHAE SANG EUN;KIM SEONG JIN;SONG HO YOUNG;PARK TAE KYO;WOO SUNG HO;KIM YONG ZU;LEE JINHWA;LEE SUK HO;LEGOCHEM BIOSCIENCE LTD.;GREEN CROSS CORPORATION 发明人 CHO YOUNG LAG;CHAE SANG EUN;KIM SEONG JIN;SONG HO YOUNG;PARK TAE KYO;WOO SUNG HO;KIM YONG ZU;LEE JINHWA;LEE SUK HO
分类号 C07D253/06 主分类号 C07D253/06
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