摘要 |
Disclosed are heterocyclic compounds, or salts thereof, represented by general formula (I). Examples of the heterocyclic compound include: N-Dimethyl-M-[6-(2-{ 4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl} -1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide, 3,4-Dichloro-N-(2-{ 2-[4-(4-isopropoxybenzyl)piperazine-1-carbonyl]-1-methyl-1H-indol-6-yloxy} pyrimidin-5-yl)-N-methylbenzenesulfonamide, and N-[6-(2-(4-[(4-Methoxybenzyl)methylamino]piperidine-1-carbonyll-1-methyl-1H-indol-5-yloxy)pyridin-3-yl]-4-trifluoromethylbenzamide. The compounds are used to treat fibrosis and tumours.
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申请人 |
OTSUKA PHARMACEUTICAL CO., LTD. |
发明人 |
SUMIDA, TAKUMI;TABUSA, FUJIO;SEKIGUCHI, KAZUO;KODAMA, TAKESHI;YASUMURA, KOICHI;KOJIMA, YUTAKA;MOTOYAMA, MASAAKI;MIYAJIMA, KEISUKE;YOSHIDA, KENJI;KAN, KEIZO;SAKAMOTO, MAKOTO;TAKASU, HIDEKI;NAKAGAWA, TAKASHI;OHI, NAOTO;HARADA, YASUO;HASHIMOTO, NORIKAZU;MATSUYAMA, HIRONORI;IIDA, MASATOSHI;FUJITA, SHIGEKAZU;FUKUSHIMA, TAE |