发明名称 HETEROCYCLIC COMPOUND AND PHARMACEUTICAL COMPOSITION THEREOF
摘要 Disclosed are heterocyclic compounds, or salts thereof, represented by general formula (I). Examples of the heterocyclic compound include: N-Dimethyl-M-[6-(2-{ 4-[4-(2,2,2-trifluoroethoxy)benzyl]piperazine-1-carbonyl} -1H-indol-6-yloxy)pyridin-3-yl]benzenesulfonamide, 3,4-Dichloro-N-(2-{ 2-[4-(4-isopropoxybenzyl)piperazine-1-carbonyl]-1-methyl-1H-indol-6-yloxy} pyrimidin-5-yl)-N-methylbenzenesulfonamide, and N-[6-(2-(4-[(4-Methoxybenzyl)methylamino]piperidine-1-carbonyll-1-methyl-1H-indol-5-yloxy)pyridin-3-yl]-4-trifluoromethylbenzamide. The compounds are used to treat fibrosis and tumours.
申请公布号 NZ584573(A) 申请公布日期 2012.05.25
申请号 NZ20080584573 申请日期 2008.10.29
申请人 OTSUKA PHARMACEUTICAL CO., LTD. 发明人 SUMIDA, TAKUMI;TABUSA, FUJIO;SEKIGUCHI, KAZUO;KODAMA, TAKESHI;YASUMURA, KOICHI;KOJIMA, YUTAKA;MOTOYAMA, MASAAKI;MIYAJIMA, KEISUKE;YOSHIDA, KENJI;KAN, KEIZO;SAKAMOTO, MAKOTO;TAKASU, HIDEKI;NAKAGAWA, TAKASHI;OHI, NAOTO;HARADA, YASUO;HASHIMOTO, NORIKAZU;MATSUYAMA, HIRONORI;IIDA, MASATOSHI;FUJITA, SHIGEKAZU;FUKUSHIMA, TAE
分类号 C07D401/12;A61K31/444;A61K31/506;A61P1/16;C07D403/12 主分类号 C07D401/12
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