发明名称 (AZA) INDOLE DERIVATIVE SUBSTITUTED IN POSITION 5, PHARMACEUTICAL COMPOSITION COMPRISING IT, INTERMEDIATE COMPOUNDS AND PREPARATION PROCESS THEREFOR
摘要 An invention refers to (aza)indole derivative substituted in position 5, of formula (I), in which X, Y, Z, G1, G2, G3, R1, W, and R2 have the meanings given in the description, which are characterized by inhibiting capabilities in respect to PGES-1, pharmaceutical compositions comprising it and a preparation process therefore.
申请公布号 GEP20125547(B) 申请公布日期 2012.05.25
申请号 GE2008AP11899 申请日期 2008.12.16
申请人 AZIENDE CHIMICHE RIUNITE ANGELINI FRANCESCO A.C.R.A.F. S.P.A. 发明人 CAZZOLLA, NICOLA;ALISI, MARIA, ALESSANDRA;FURLOTTI, GUIDO;MANGANO, GIORGINA;COLETTA, ISABELLA;MAUGER, CATERINA;DRAGONE, PATRIZIA;GAROFALO, BARBARA;GARRONE, BEATRICE
分类号 C07D209/08;A61K31/404;A61K31/437;C07D209/12;C07D209/18;C07D401/04;C07D471/04 主分类号 C07D209/08
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