发明名称 Heterocyclic compounds as factor IXA inhibitors
摘要 The present invention relates to novel heterocyclic compounds of Formulae I-III; as disclosed herein or a pharmaceutically acceptable salt, solvate, ester, prodrug or stereoisomer thereof. Also disclosed are pharmaceutical compositions comprising said compounds, and methods for using said compounds for treating or preventing a thromboembolic disorder.
申请公布号 US8148363(B2) 申请公布日期 2012.04.03
申请号 US20090993607 申请日期 2009.05.18
申请人 CLASBY MARTIN C.;GREENLEE WILLIAM J.;XIA YAN;CHAN TIN-YAU;CHELLIAH MARIAPPAN V.;CHACKALAMANNIL SAMUEL;PU HAIYAN;EAGEN KEITH A.;VACCARO HENRY;MCKITTRICK BRIAN A.;WANG LIYUAN;GAO XIAOBANG;SCHERING CORPORATION 发明人 CLASBY MARTIN C.;GREENLEE WILLIAM J.;XIA YAN;CHAN TIN-YAU;CHELLIAH MARIAPPAN V.;CHACKALAMANNIL SAMUEL;PU HAIYAN;EAGEN KEITH A.;VACCARO HENRY;MCKITTRICK BRIAN A.;WANG LIYUAN;GAO XIAOBANG
分类号 A61K31/55;A61K31/4184;A61K31/4192;A61K31/422;A61K31/4439;A61K31/454;A61K31/496;A61K31/506;A61K31/5377;A61P7/02;C07D401/14;C07D403/04;C07D403/14;C07D413/14 主分类号 A61K31/55
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