发明名称 |
Heterocyclic compounds as factor IXA inhibitors |
摘要 |
The present invention relates to novel heterocyclic compounds of Formulae I-III; as disclosed herein or a pharmaceutically acceptable salt, solvate, ester, prodrug or stereoisomer thereof. Also disclosed are pharmaceutical compositions comprising said compounds, and methods for using said compounds for treating or preventing a thromboembolic disorder. |
申请公布号 |
US8148363(B2) |
申请公布日期 |
2012.04.03 |
申请号 |
US20090993607 |
申请日期 |
2009.05.18 |
申请人 |
CLASBY MARTIN C.;GREENLEE WILLIAM J.;XIA YAN;CHAN TIN-YAU;CHELLIAH MARIAPPAN V.;CHACKALAMANNIL SAMUEL;PU HAIYAN;EAGEN KEITH A.;VACCARO HENRY;MCKITTRICK BRIAN A.;WANG LIYUAN;GAO XIAOBANG;SCHERING CORPORATION |
发明人 |
CLASBY MARTIN C.;GREENLEE WILLIAM J.;XIA YAN;CHAN TIN-YAU;CHELLIAH MARIAPPAN V.;CHACKALAMANNIL SAMUEL;PU HAIYAN;EAGEN KEITH A.;VACCARO HENRY;MCKITTRICK BRIAN A.;WANG LIYUAN;GAO XIAOBANG |
分类号 |
A61K31/55;A61K31/4184;A61K31/4192;A61K31/422;A61K31/4439;A61K31/454;A61K31/496;A61K31/506;A61K31/5377;A61P7/02;C07D401/14;C07D403/04;C07D403/14;C07D413/14 |
主分类号 |
A61K31/55 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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