发明名称 SUBSTITUTED AMINO - BENZOIC ACID DERIVATIVES AS INHIBITORS OF DNA METHYLTRANSFERASES
摘要 <p>The present invention relates to a compound having the following formula (I), wherein : - R1 and R2 are alkyl groups having from 1 to 12 carbon atoms; - X1 is NH or O;- R3, R4, R5 and R6 are in particular H; - X2 is in particular -CH2-; - n is an integer comprised from 2 to 20; and - R is an inhibitor of DNA methyltransferases, or its pharmaceutically acceptable salts, hydrates or hydrated salts or its polymorphic crystalline structures, racemates, diastereomers or enantiomers.</p>
申请公布号 WO2012038417(A1) 申请公布日期 2012.03.29
申请号 WO2011EP66305 申请日期 2011.09.20
申请人 INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM);CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S);MUSEUM NATIONAL D'HISTOIRE NATURELLE;GUIANVARC'H, DOMINIQUE;ARIMONDO, PAOLA;SENAMAUD-BEAUFORT, CATHERINE;GRELLIER, PHILIPPE;HALBY, LUDOVIC;FERROUD, CLOTILDE;CNAM CONSERVATOIRE NATIONAL DES ARTS DES METIERS 发明人 GUIANVARC'H, DOMINIQUE;ARIMONDO, PAOLA;SENAMAUD-BEAUFORT, CATHERINE;GRELLIER, PHILIPPE;HALBY, LUDOVIC;FERROUD, CLOTILDE
分类号 C07D209/48;A61K31/4035;A61P25/00;A61P33/00;A61P35/00;C07D311/30;C07D403/06 主分类号 C07D209/48
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