摘要 |
<p>The present invention relates to a compound having the following formula (I), wherein : - R1 and R2 are alkyl groups having from 1 to 12 carbon atoms; - X1 is NH or O;- R3, R4, R5 and R6 are in particular H; - X2 is in particular -CH2-; - n is an integer comprised from 2 to 20; and - R is an inhibitor of DNA methyltransferases, or its pharmaceutically acceptable salts, hydrates or hydrated salts or its polymorphic crystalline structures, racemates, diastereomers or enantiomers.</p> |
申请人 |
INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE (INSERM);CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S);MUSEUM NATIONAL D'HISTOIRE NATURELLE;GUIANVARC'H, DOMINIQUE;ARIMONDO, PAOLA;SENAMAUD-BEAUFORT, CATHERINE;GRELLIER, PHILIPPE;HALBY, LUDOVIC;FERROUD, CLOTILDE;CNAM CONSERVATOIRE NATIONAL DES ARTS DES METIERS |
发明人 |
GUIANVARC'H, DOMINIQUE;ARIMONDO, PAOLA;SENAMAUD-BEAUFORT, CATHERINE;GRELLIER, PHILIPPE;HALBY, LUDOVIC;FERROUD, CLOTILDE |