发明名称 |
ANTAGONISTAS DEL RECEPTOR HISTAMINA H3. |
摘要 |
Un compuesto seleccionado entre: 5-(4-clorofenil)-2-(4-isopropilpiperacin-1-il)pirimidina; 2-(4-isopropilpiperacin-1-il)-5-(4-trifluorometilfenil)pirimidina; 4-[2-(4-isopropilpiperacin-1-5 il)pirimidin-5-il]benzonitrilo; 5-(4-fluorofenil)-2-(4-isopropilpiperacin-1-il)pirimidina; 2-(4-isopropilpiperacin-1-il)-5-(4-trifluorometoxilfenil)pirimidina; 2-(4-isopropilpiperacin-1-il)-5-(4-metoxilfenil)pirimidina; 4-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]benzonitrilo; N-{4-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]bencil}acetamida; {4-[2-(4-isopropilpiperacin-1-il)pirimidin-6-il]fenil}acetonitrilo; N-{4-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]fenil}acetamida; 1-{4-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]fenil}etanona; 2-(4-isopropilpiperacin-1-il)-5-piridin-3-ilpirimidina; 2-(4-isopropilpiperacin-1-il)-5-piridin-4-ilpirimidina; {4-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]fenil}dimetilamina; 3-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]-N,N-dimetilbenzamida; 4-{4-[2-(4-ciclopropilpiperacin-1-il)pirimidin-5-il]bencil}morfolina; N-{4-[2-(4-isopropilpiperacin-1-il)pirimidin-5-il]bencil}isobutiramida; 4-[2-(4-ciclopropilpiperacin-1-il)pirimidin-5-il]bencilamina; y N-{4-[2-(4-ciclopropilpiperacin-1-il)pirimidin-5-il]bencil}acetamida; o una sal o solvato aceptable farmacéuticamente de las mismas.
|
申请公布号 |
ES2375929(T3) |
申请公布日期 |
2012.03.07 |
申请号 |
ES20100166493T |
申请日期 |
2006.06.30 |
申请人 |
HIGH POINT PHARMACEUTICALS, LLC |
发明人 |
HOHLWEG, ROLF;ANDERSEN, KNUD ERIK;SOERENSEN, JAN LINDY;LUNDBECK, JANE MARIE |
分类号 |
C07D213/74;A61K31/444;A61P3/00;C07D213/84;C07D213/87;C07D241/20;C07D401/04;C07D401/08;C07D401/12;C07D403/04;C07D403/12;C07D405/06;C07D413/04;C07D413/10;C07D413/14 |
主分类号 |
C07D213/74 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|