发明名称 |
BICYCLOESTER DERIVATIVE |
摘要 |
<p>SUMMARY Novel bicycloester derivatives and pharmaceutically acceptable salts thereof have high DPP-IV inhibitory activity. SOLVING MEANS The novel bicycloester derivatives are represented by the general formula (1):
Pharmaceutically acceptable salts thereof are also included (Example: (2S,4S)-1-[[N-(4-ethoxycarbonylbicyclo[2.2.2]oct-1-yl)amino]acetyl]-4-fluoropyrrolidine-2-carbonitrile)).</p> |
申请公布号 |
PT1712547(E) |
申请公布日期 |
2012.03.06 |
申请号 |
PT20050704327T |
申请日期 |
2005.02.01 |
申请人 |
KYORIN PHARMACEUTICAL CO., LTD. |
发明人 |
YASUMICHI FUKUDA;YOSHIKAZU ASAHINA;KOHEI OHATA;KAZUYA YOKOTA;TOSHIYUKI MATSUI |
分类号 |
C07D207/16;A61K31/40;A61K31/4025;A61P3/10;A61P43/00;C07D405/12 |
主分类号 |
C07D207/16 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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