发明名称 |
Substituted piperidines as Par-1 Antagonists |
摘要 |
The invention relates to novel substituted piperidines, to processes for their preparation, to their use for the treatment and/or prophylaxis of diseases and to their use for preparing medicaments for the treatment and/or prophylaxis of diseases, in particular of cardiovascular disorders and tumour disorders.
|
申请公布号 |
US2012046268(A1) |
申请公布日期 |
2012.02.23 |
申请号 |
US201013202707 |
申请日期 |
2010.03.12 |
申请人 |
JESKE MARIO;HEIMBACH DIRK;ROEHRIG SUSANNE;CANCHO GRANDE YOLANDA;SCHNEIDER DIRK;RESTER ULRICH;BENDER ECKHARD;MEININGHAUS MARK;ZIMMERMANN KATJA;ZUBOV DMITRY;BUCHMUELLER ANJA;VON DEGENFELD GEORGES;GERDES CHRISTOPH;GERISCH MICHAEL;GNOTH MARK JEAN;GERICKE KERSTEN MATTHIAS;BAYER PHARMA AKTIENGESELLSCHAFT |
发明人 |
JESKE MARIO;HEIMBACH DIRK;ROEHRIG SUSANNE;CANCHO GRANDE YOLANDA;SCHNEIDER DIRK;RESTER ULRICH;BENDER ECKHARD;MEININGHAUS MARK;ZIMMERMANN KATJA;ZUBOV DMITRY;BUCHMUELLER ANJA;VON DEGENFELD GEORGES;GERDES CHRISTOPH;GERISCH MICHAEL;GNOTH MARK JEAN;GERICKE KERSTEN MATTHIAS |
分类号 |
A61K31/4523;A61K31/445;A61K31/4525;A61K31/453;A61K31/454;A61K31/4545;A61K31/496;A61K31/5377;A61K31/541;A61P7/02;C07D211/60;C07D401/06;C07D405/06;C07D413/06;C07D417/06;C12N5/078 |
主分类号 |
A61K31/4523 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|