发明名称 |
LHRH-II PEPTIDE ANALOGS |
摘要 |
The invention is directed to analogs of LHRH-II and, more generally, to analogs of the LHRH family in which modifications have been made that confer enhanced binding affinity for LHRH receptors and/or improved metabolic stability. The invention is further directed to methods of targeted therapy and targeted imaging in patients with sex-hormone-related cancers or other LHRH-mediated diseases.
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申请公布号 |
US2012045393(A1) |
申请公布日期 |
2012.02.23 |
申请号 |
US201013256912 |
申请日期 |
2010.03.16 |
申请人 |
LINDER KAREN E.;NANJAPPAN PALANIAPPA;RAJU NATARAJAN;KHURANA SUDHA;SWENSON ROLF E.;NUNN ADRIAN D.;RAMALINGAM KONDAREDDIAR |
发明人 |
LINDER KAREN E.;NANJAPPAN PALANIAPPA;RAJU NATARAJAN;KHURANA SUDHA;SWENSON ROLF E.;NUNN ADRIAN D.;RAMALINGAM KONDAREDDIAR |
分类号 |
A61K49/00;A61K38/08;A61K38/09;A61K49/04;A61K49/14;A61K49/22;A61K51/08;A61P35/00;C07K7/06;C07K7/23 |
主分类号 |
A61K49/00 |
代理机构 |
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代理人 |
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地址 |
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