发明名称 |
Preparation of C-Pyrazine-Methylamines |
摘要 |
A process for preparing a compound of formula (I) or a salt thereof: (I) wherein R1 is H or optionally substituted aryl or heteroaryl; comprising reacting 2,3-dichloropyrazine with a suitable diaryl imine followed by hydrolysis.
|
申请公布号 |
US2012041202(A1) |
申请公布日期 |
2012.02.16 |
申请号 |
US201013265363 |
申请日期 |
2010.04.19 |
申请人 |
MAO YUNYU;MULVIHILL KRISTEN MICHELLE;RECHKA JOSEF A.;TAVARES-GRECO PAULA A.;OSI PHARMACEUTICALS, LLC |
发明人 |
MAO YUNYU;MULVIHILL KRISTEN MICHELLE;RECHKA JOSEF A.;TAVARES-GRECO PAULA A. |
分类号 |
C07D487/04;C07D241/16;C07D401/10 |
主分类号 |
C07D487/04 |
代理机构 |
|
代理人 |
|
主权项 |
|
地址 |
|