发明名称 SULFONYLAMINO-DERIVATIVES, COMPOSITIONS THEREOF, PROCESS OF PREPARATION AND USES FOR THE MANUFACTURE OF MEDICAMENTS FOR INHIBITING HISTONE DEACETYLASE
摘要 This invention comprises the novel compounds of formula (I) wherein n, m, t, R1, R2, R3, R4, R5, L, Q, X, Y, Z and have defined meanings, having histone deacetylase inhibiting enzymatic activity; their preparation, compositions containing them and their use as a medicine.
申请公布号 IL164003(A) 申请公布日期 2011.12.29
申请号 IL20040164003 申请日期 2004.09.09
申请人 JANSSEN PHARMACEUTICAL, N.V. 发明人
分类号 C07D239/42;A61K31/40;A61K31/4025;A61K31/438;A61K31/4427;A61K31/445;A61K31/451;A61K31/4545;A61K31/472;A61K31/495;A61K31/496;A61K31/497;A61K31/506;A61K31/517;A61K31/53;A61K31/5377;A61K31/55;A61K31/551;A61K45/00;A61P1/04;A61P1/18;A61P3/10;A61P5/00;A61P9/00;A61P9/02;A61P9/08;A61P9/10;A61P11/00;A61P11/02;A61P11/06;A61P13/08;A61P13/10;A61P13/12;A61P15/00;A61P17/00;A61P17/04;A61P17/06;A61P17/10;A61P17/14;A61P17/16;A61P19/00;A61P19/02;A61P19/06;A61P21/04;A61P25/00;A61P25/16;A61P25/28;A61P27/02;A61P27/06;A61P29/00;A61P31/18;A61P35/00;A61P35/02;A61P37/02;A61P37/04;A61P37/06;A61P37/08;A61P43/00;C07D207/09;C07D207/14;C07D211/26;C07D211/58;C07D213/74;C07D213/78;C07D217/02;C07D217/04;C07D241/04;C07D249/12;C07D295/14;C07D295/155;C07D295/20;C07D295/22;C07D295/26;C07D307/68;C07D317/58;C07D401/04;C07D401/06;C07D401/12;C07D401/14;C07D403/04;C07D403/12;C07D405/12;C07D405/14;C07D409/12;C07D409/14;C07D413/02;C07D413/04;C07D413/12;C07D471/10;C12Q1/48 主分类号 C07D239/42
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