METHODS AND COMPOUNDS FOR THE PREPARATION OF MONOFLUOROMETHYLATED BIOLOGICALLY ACTIVE ORGANIC COMPOUNDS
摘要
<p>The present invention describes processes for the preparation of, monofluoromethylated organic biologically active compounds, such as Fluticasone Propionate and Fluticasone Furoate, in the presence of fluorodecarboxylating reagents such as XeF2 and BrF3.</p>
申请公布号
WO2011151625(A1)
申请公布日期
2011.12.08
申请号
WO2011GB00835
申请日期
2011.06.01
申请人
HOVIONE INTER LIMITED;LEITAO, EMILIA, PERPETUA, TAVARES;HEGGIE, WILLIAM;TURNER, CRAIG, ROBERT