发明名称 |
PYRANONE COMPOUNDS USEFUL TO TREAT RETROVIRAL INFECTIONS |
摘要 |
The present invention relates to compounds of formula I and II which are pyran-2-ones, 5,6-dihydro-pyran-2-ones, 4-hydroxy-benzopyran-2-ones, 4-hydroxy-cycloalkyl[b]pyran-2-ones, and derivatives thereof, useful for inhibiting a retrovirus in a mammalian cell infected with said retrovirus.wherein R10 and R20 taken together are: |
申请公布号 |
HK1084667(A1) |
申请公布日期 |
2011.12.02 |
申请号 |
HK20060104885 |
申请日期 |
2006.04.25 |
申请人 |
PHARMACIA & UPJOHN COMPANY |
发明人 |
KAREN RENE ROMINES;GORDON L. BUNDY;THERESA M. SCHWARTZ;RUBEN A. TOMMASI;JOSEPH WALTER STROHBACH;STEVEN RONALD TURNER;SUVIT THAISRIVONGS;PAUL ADRIAN ARISTOFF;PAUL D. JOHNSON;HARVEY IRVING SKULNICK;LOUIS L. SKALETZKI;DAVID JOHN ANDERSON;JOEL MORRIS;RONALD B. GAMMILL;GEORGE P. LUKE |
分类号 |
A61K31/365;A61K31/366;A61K31/415;A61K31/425;A61K31/44;A61K31/4427;A61K31/443;A61K31/47;A61K31/4709;A61K31/505;A61K31/506;A61K31/54;A61P31/12;C07D;C07D309/32;C07D309/38;C07D309/40;C07D311/02;C07D311/08;C07D311/74;C07D311/94;C07D401/12;C07D403/12;C07D405/00;C07D405/12;C07D405/14;C07D407/00;C07D409/00;C07D417/00;C07D417/12 |
主分类号 |
A61K31/365 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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