发明名称 |
2,4-DIOXO-1,4-DIHYDRO-2H-QUINAZOLIN-3-YL-SULFONAMIDE DERIVATIVES |
摘要 |
<p>The invention relates to a 2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl-sulfonamide derivative being (A) a compound of the formula (I) in which the substituents are as defined in the specification; in free form or in salt form; or (B) a compound selected from a certain group of 2,4-dioxo-1,4-dihydro-2H-quinazolin-3-yl-sulfonamide derivatives disclosed in the specification; in free form or in salt form; to their preparation, to their use as medicament and to medicaments comprising them. In a first aspect, the invention provides prodrugs of AMPA receptor antagonists which potentially useful in the treatment of a wide range of disorders, particularly epilepsy.</p> |
申请公布号 |
WO2011144666(A1) |
申请公布日期 |
2011.11.24 |
申请号 |
WO2011EP58068 |
申请日期 |
2011.05.18 |
申请人 |
NOVARTIS AG;AUBERSON, YVES;CARCACHE, DAVID;LERCHNER, ANDREAS;NOZULAK, JOACHIM |
发明人 |
AUBERSON, YVES;CARCACHE, DAVID;LERCHNER, ANDREAS;NOZULAK, JOACHIM |
分类号 |
C07D403/04;A61K31/517;A61P25/08;C07D405/04 |
主分类号 |
C07D403/04 |
代理机构 |
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代理人 |
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主权项 |
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地址 |
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